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所有目前已知的FGFR1、2、3、4突变率
所有目前已知的FGFR1、2、3、4突变率
行业数据
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图片格式:PNG
图片大小:779KB
图片尺寸:1194*969
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所属报告:
诺诚健华~B-Biotech新秀崛起重塑BTK大市场新格局-210718(35页).pdf
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相关数据
anti-FGFR2b单抗与SOS1抑制剂国内临床进展
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行业数据
2025-12-31
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图表30FGFR4与FGFR1-3结构差异
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行业数据
2025-04-11
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FGFR4不同于FGFR1-3(LoopIIIb和LoopIIIc),仅有LoopIIIc
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行业数据
2022-08-24
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中国主要FGFR1/2/3畸变癌症新发病例
fCDlubTku70gfCDkubPohbrnmYzvvIjljYPkvovvvIkgfCDog4PnmYzvvIjljYPkvovvvIkgfCDog4bnrqHnmYzvvIjljYPkvovvvIkgfCDlsL/ot6/kuIrnmq7nmYzvvIjljYPkvovvvIkgfAp8LS0tLS0tfC0tLS0tLS0tLS0tLS0tLS18LS0tLS0tLS0tLS0tLS18LS0tLS0tLS0tLS0tLS0tLXwtLS0tLS0tLS0tLS0tLS0tLS18CnwgMjAxNiB8IDU0ICAgICAgICAgICAgIHwgMjggICAgICAgICAgIHwgMjYgICAgICAgICAgICAgfCAyMiAgICAgICAgICAgICAgIHwKfCAyMDIwIHwgNTggICAgICAgICAgICAgfCAzMSAgICAgICAgICAgfCAyOSAgICAgICAgICAgICB8IDI0ICAgICAgICAgICAgICAgfAp8IDIwMjVFfCA2MiAgICAgICAgICAgICB8IDM3ICAgICAgICAgICB8IDM0ICAgICAgICAgICAgIHwgMjkgICAgICAgICAgICAgICB8CnwgMjAzMEV8IDY1ICAgICAgICAgICAgIHwgNDIgICAgICAgICAgIHwgNDAgICAgICAgICAgICAgfCAzNCAgICAgICAgICAgICAgIHwKfCAyMDM1RXwgNjcgICAgICAgICAgICAgfCA0NiAgICAgICAgICAgfCA0NSAgICAgICAgICAgICB8IDM4ICAgICAgICAgICAgICAgfAoK6LWE5paZ5p2l5rqQ77yaRnJvc3QgJiBTdWxsaXZhbuOAgea1pumTtuWbvemZhQ==
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行业数据
2022-08-02
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中国主要FGFR1/2/3畸变癌症新发病例
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行业数据
2022-08-01
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国内处于临床阶段的泛FGFR抑制剂和FGFR1/2/3抑制剂
<table border="1" cellspacing="0" cellpadding="5">
    <thead>
        <tr style="background-color: #004080; color: white;">
            <th>药物名称</th>
            <th>公司名称</th>
            <th>适应症</th>
            <th>临床阶段</th>
            <th>首次公示日期</th>
        </tr>
    </thead>
    <tbody>
        <tr>
            <td rowspan="3">Pemigatinib</td>
            <td rowspan="3">信达</td>
            <td>一线胆管癌</td>
            <td>递交上市申请</td>
            <td>2021/7/2</td>
        </tr>
        <tr>
            <td>二线胆管癌</td>
            <td>二期</td>
            <td>2019/12/27</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2019/12/23</td>
        </tr>
        <tr>
            <td rowspan="5">Erdafitinib</td>
            <td rowspan="5">强生</td>
            <td>二线尿路上皮癌</td>
            <td>三期</td>
            <td>2018/11/27</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>二期</td>
            <td>2017/7/5</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>二期</td>
            <td>2020/3/23</td>
        </tr>
        <tr>
            <td>非肌层浸润性膀胱肿瘤</td>
            <td>二期</td>
            <td>2020/9/15</td>
        </tr>
        <tr>
            <td>二线晚期肝细胞癌</td>
            <td>I/II期</td>
            <td>2017/7/25</td>
        </tr>
        <tr>
            <td rowspan="2">Infigratinib</td>
            <td rowspan="2">Alcami</td>
            <td>胆管癌</td>
            <td>三期</td>
            <td>2021/2/18</td>
        </tr>
        <tr>
            <td>胃癌或胃食管结合部腺癌</td>
            <td>二期</td>
            <td>2021/2/25</td>
        </tr>
        <tr>
            <td rowspan="3">HMPL - 453</td>
            <td rowspan="3">和黄医药</td>
            <td>晚期恶性复治间皮瘤</td>
            <td>二期</td>
            <td>2019/11/4</td>
        </tr>
        <tr>
            <td>晚期肝内胆管癌</td>
            <td>二期</td>
            <td>2020/5/22</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>I/II期</td>
            <td>2017/7/28</td>
        </tr>
        <tr>
            <td rowspan="2">ICP - 192</td>
            <td rowspan="2">诺诚健华</td>
            <td>尿路上皮癌</td>
            <td>二期</td>
            <td>2020/4/27</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>I/II期</td>
            <td>2018/11/22</td>
        </tr>
        <tr>
            <td>E7090</td>
            <td>卫材</td>
            <td>胆管癌</td>
            <td>二期</td>
            <td>2020/8/14</td>
        </tr>
        <tr>
            <td>Derazantinib</td>
            <td>仑胜医药</td>
            <td>胆管癌</td>
            <td>I/II期</td>
            <td>2019/5/27</td>
        </tr>
        <tr>
            <td rowspan="4">AL 8326</td>
            <td rowspan="4">爱德程医药</td>
            <td>小细胞肺癌</td>
            <td>I/II期</td>
            <td>2020/9/11</td>
        </tr>
        <tr>
            <td>妇科恶性肿瘤</td>
            <td>一期</td>
            <td>2021/1/18</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2018/12/12</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2017/2/3</td>
        </tr>
        <tr>
            <td rowspan="3">MAX 40279</td>
            <td rowspan="3">再极医药</td>
            <td>MDS，复发或难治性 AML</td>
            <td>I/II期</td>
            <td>2021/6/2</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2019/12/26</td>
        </tr>
        <tr>
            <td>复发难治性 AML</td>
            <td>一期</td>
            <td>2019/10/9</td>
        </tr>
        <tr>
            <td>BGJ398</td>
            <td>诺华</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2014/9/11</td>
        </tr>
        <tr>
            <td>EOC317</td>
            <td>亿腾景昂</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2018/4/9</td>
        </tr>
        <tr>
            <td>HH185</td>
            <td>上海海和、思路迪</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2018/10/23</td>
        </tr>
        <tr>
            <td>SYHA1803</td>
            <td>石药</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2019/6/28</td>
        </tr>
        <tr>
            <td>SC0011</td>
            <td>智康弘仁</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2021/2/18</td>
        </tr>
        <tr>
            <td>BPI - 17509</td>
            <td>贝达药业</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2019/10/23</td>
        </tr>
        <tr>
            <td rowspan="2">AL58805</td>
            <td rowspan="2">爱德程医药</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2021/4/15</td>
        </tr>
        <tr>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2019/1/14</td>
        </tr>
        <tr>
            <td>AZD 4547</td>
            <td>和誉生物</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2021/4/23</td>
        </tr>
        <tr>
            <td>HZB1006</td>
            <td>哈尔滨珍宝</td>
            <td>晚期实体瘤</td>
            <td>一期</td>
            <td>2021/5/25</td>
        </tr>
    </tbody>
</table>

<p>资料来源：丁香园，申万宏源研究</p>
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2021-08-18
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ICP-192对FGFR1-4的抑制作用和erdafitinib
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2021-08-18
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尿道上皮癌(UC)、胆管癌(CCA)突变率高,临床存在较大未满足需求。成纤维细胞生长因子受体(FGFR)是高度保守及高表达的跨膜酪氨酸激酶受体。FGFR 是高度相似受体家族,包括 FGFR 1-4。FGFR 异常于实体瘤患者中常见,占所有实体瘤患者约 7.1%。FGFR 抑制剂通过与FGFR1-4 的 ATP 结合位点不可逆地共价结合,抑制 FGFR 介导的信号传导,从而降低携带 FGFR1-4 基因变异的肿瘤细胞的增殖。最常受FGFR 异常影响的癌症包括尿道上皮癌(31 .7%)、胆管癌(25.2%)、肝细胞癌(20 .0%)、乳癌(17 .5%)及胃癌(6 .7%)。其中 UC 是中国第九种最常见的癌症,也是男性癌症病例中第七大病因。UC 经常复发,化疗仍然是 UC 的标准治疗方法。胆管癌(CCA)是一种沿着胆管形成的癌症,属罕见的恶性肿瘤,死亡率高,就晚期患者而言,现时疗法对整体存活率并无重大改善。因此对于此两种疾病的新疗法开发具有十分重要的意义。公司正积极推动 ICP-192 的针对 CCA 及 UC 的临床试验。
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