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EGFRTKI突变机理及占比
EGFRTKI突变机理及占比
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所属报告:
【公司研究】贝达药业-多款产品即将上市自主研发逐步验证-210316(45页).pdf
打包全文图表
相关数据
图23.2024年国内EGFRTKI市场份额
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竞争格局
2026-01-13
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图表11国内EGFRTKI样本医院销售额/及
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行业数据
2025-12-03
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图11.中国三代EGFRTKI竞争格局
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竞争格局
2025-06-17
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三代EGFRTKI药物获批和医保目录纳入情况
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行业数据
2025-06-09
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2020-2024年三代EGFRTKI样本医院销售金额占比
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行业数据
2025-06-09
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2020-2024年各代EGFRTKI样本医院销售金额占比
fCDlubTku70gfCDnrKzkuIDku6MgfCDnrKzkuozku6MgfCDnrKzkuInku6MgfAp8LS0tLS0tfC0tLS0tLS0tfC0tLS0tLS0tfC0tLS0tLS0tfAp8IDIwMjAgfCA1OCUgICAgfCAwJSAgICAgfCAwJSAgICAgfAp8IDIwMjEgfCA2MyUgICAgfCAwJSAgICAgfCAwJSAgICAgfAp8IDIwMjIgfCA3NCUgICAgfCAwJSAgICAgfCAwJSAgICAgfAp8IDIwMjMgfCA3NiUgICAgfCAwJSAgICAgfCAwJSAgICAgfAp8IDIwMjQgfCA3OSUgICAgfCAwJSAgICAgfCAwJSAgICAgfAoK6LWE5paZ5p2l5rqQ77ya5Yy76I2v6a2U5pa577yM5aSp6aOO6K+B5Yi456CU56m25omA
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行业数据
2025-06-09
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三代EGFRTKI奥希替尼历年全球销售额
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行业数据
2025-04-18
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截至2025年2月,多款针对EGFRTKI耐药后NSCLC患者(全人群)的药物全球进度较快
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行业数据
2025-04-14
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中国EGFRTKI销售情况(亿元)
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行业数据
2025-03-03
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图表13国内已上市第三代EGFRTKI临床数据
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行业数据
2025-02-24
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图表67我国一二三代EGFRTKI市占率
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竞争格局
2025-02-24
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EGFRTKI对Exon20ins和敏感突变的敏感度
fCBUS0kgfCBFeG9uMjBpbnPmlY/mhJ/luqbovoNMODU4UuS9jiB8CnwtLS0tLS18LS0tLS0tLS0tLS0tLS0tLS0tLS0tLS0tLS18CnwgMeS7oyAgfCA+MTk05YCNICAgICAgICAgICAgICAgICAgIHwKfCAy5LujICB8IDQ1LTE1NeWAjSAgICAgICAgICAgICAgICAgfAp8IDPku6MgIHwgMTEtOTTlgI0gICAgICAgICAgICAgICAgICB8CgrotYTmlpnmnaXmupDvvJrlhazlj7jlrpjnvZHvvIzkuJzlkLTor4HliLjnoJTnqbbmiYA=
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行业数据
2025-02-06
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第三代EGFRTKI大部分为苯胺基嘧啶类衍生物
5oqx5q2J77yM5oiR5peg5rOV5o+Q5Y+W5Zu+54mH5Lit55qE5pWw5o2u5oiW55Sf5oiQ6KGo5qC844CC6K+35oKo5o+Q5L6b5paH5a2X5o+P6L+w5oiW5YW25LuW5L+h5oGv77yM5oiR5Lya5bC95Yqb5biu5Yqp5oKo44CC
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行业数据
2025-01-16
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截至2024年11月,我国已获批6款第三代EGFRTKI
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行业数据
2025-01-16
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我国EGFRTKI市场规模不断增长(亿元)
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市场规模
2025-01-16
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其中约 60%的患者 EGFR T790M 突变。突变产生的空间位阻将阻碍一代、二代 TKI 结合,从而产生耐药性。三代 EGFR TKI 例如奥希替尼采用嘧啶母环可克服 T790M 产生的空间位阻,从而克服患者的耐药性。因此,三代 EGFR TKI可用于经一、二代产品治疗后耐药患者。
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