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图表10伊布替尼、泽布替尼和奥布替尼国内纳入医保情况
图表10伊布替尼、泽布替尼和奥布替尼国内纳入医保情况
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诺诚健华-公司研究报告-始于创新、强于执行力血液瘤及自免领域管线双开花-240321(38页).pdf
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一线CLL/SLL诊疗指南:泽布替尼为首选推荐(PreferredRegiments)用药
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行业数据
2025-08-07
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一线CLL/SLL持续治疗方案III期临床数据(非头对头对比):泽布替尼展现同类最优潜力
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行业数据
2025-08-07
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BTK抑制剂全球销售额(百万美元):泽布替尼市场份额持续攀升
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竞争格局
2025-08-07
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2019Q4-2025Q1泽布替尼在中国、美国的销售额(单位:百万美元)
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行业数据
2025-07-23
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图8奥雷巴替尼临床获益以及耐受性情况
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行业数据
2025-06-30
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图9奥雷巴替尼临床获益以及耐受性情况(续)
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行业数据
2025-06-30
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图11奥雷巴替尼在Ph+ALL适应症的临床疗效(续)
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2025-06-30
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图7奥雷巴替尼(HQP1351)临床推进情况
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2025-06-30
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r/rWM临床数据:泽布替尼vs伊布替尼(ASPEN研究)
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2025-06-25
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泽布替尼为同类最佳BTK抑制剂
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2025-04-18
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泽布替尼美国/中国历年销售拆分
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2025-04-18
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2026-07-30
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国内三款 BTK抑制剂(伊布替尼、泽布替尼、奥布替尼)均已进入医保,奥布替尼年治疗费用相较最低。2017年伊布替尼国内上市,当年纳入医保,降价 65%左右,医保支付价格 189元/粒/140mg;2020年泽布替尼国内上市,当年纳入医保,降价 44%左右,医保支付价在 99元/粒/80mg,2021年新增WM适应症,续约谈判价格为85元/粒/80mg(在 2020年基础上再度降价 14%)。2020年底奥布替尼国内上市,2021年公司采取的销售策略为赠药模式,2021年底进入医保目录后取消赠药,医保支付价为 119元/粒/50mg,降幅 51%左右,2023年奥布替尼新增 2L MZL适应症,最新医保价格较 2023年未降低。从治疗费用来看,奥布替尼相比进口伊布替尼具备价格优势,略低于泽布替尼。
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诺诚健华-公司研究报告-始于创新、强于执行力血液瘤及自免领域管线双开花-240321(38页).pdf
图表9第一二代BTK抑制剂结合BTK的半胱氨酸481残基(C481)
图表8全球获批上市第一二三代BTKi对比
图表7BTK信号通路
图表66参数假设及公司估值
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