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EGFR外显子20突变在EGFR相关罕见突变中占比高
EGFR外显子20突变在EGFR相关罕见突变中占比高
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图片大小:878KB
图片尺寸:1730*780
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所属报告:
和誉:专注小分子肿瘤治疗打造差异化产品-220823(43页).pdf
打包全文图表
相关数据
SHR-A2009用于EGFR突变型NSCLC的1期临床研究结果
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行业数据
2026-05-28
原图定位
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Ph2a临床研究Sefaxersen尿蛋白及eGFR数据
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行业数据
2026-03-13
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Ph3NeflgArd研究第24个月eGFR及uPCR数据
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行业数据
2026-03-13
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Ph1/2ADU-CL-19研究中Zigakibart组受试者100周uPCR及eGFR数据
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行业数据
2026-03-13
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Ph1/2aRUBY-3研究中Povetacicept80mg剂量组第48周uPCR及eGFR数据
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行业数据
2026-03-13
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图3 mCRC中EGFR抑制剂的美国收入(2004-2017)
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2026-02-13
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三代EGFR药物适应症对比(2025年新增两款)
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行业数据
2026-02-04
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第二代EGFR-TKI不同企业竞争格局
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竞争格局
2026-01-08
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第一代EGFR-TKI不同企业竞争格局
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竞争格局
2026-01-08
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Iza-bren已开展临床研究的癌种(左图中以红字标明)以及EGFR和HER3在各种上皮肿瘤中的
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行业数据
2025-12-26
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EGFR/HER3ADC全球格局
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竞争格局
2025-12-26
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图表20EGFR耐药后NSCLC试验数据比
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行业数据
2025-12-03
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和誉ABSK043的临床定位以及未来结合EGFR/KRAS等小分子抑制剂在NSCLC中布局的管线矩阵
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行业数据
2025-10-10
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EGFR突变NSCLC患者推荐用药(CSCO及NCCN指南)
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行业数据
2025-09-23
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截至2025年9月,全球共6款EGFR单抗ADC药物进入临床
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行业数据
2025-09-23
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全球拥有AKK专利菌株的核心企业
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2026-07-30
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EGFR属于一种蛋白质,是表皮生长因子的细胞表面受体酪氨酸激酶。 EGFR的活化可导致一系列下游信号活性,从而激活肿瘤细胞生长、存活、入侵、转移及抑制细胞凋亡。因此,一般认为EGFR家族的突变及失调与各种癌症有关。NSCLC是最常见的肺癌类型,约占病例的 85% 。约 10% 的 NSCLC 患者有 EGFR 外显子 20插入突变(EGFR20ins)。由于EGFR20ins结构上存在空间位阻效应,对第一/二/三代 EGFR TKI的治疗缺乏反应,目前的一线治疗策略仍然是以铂类为基础的标准化疗,但该治疗方案总体预后欠佳,中位生存时间(约16个月)明显短于经典EGFR突变(3年左右),EGFR20ins NSCLC仍然是EGFR通路上的治疗难点。
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