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PEG修饰脂质体在mRNA疫苗领域的应用
PEG修饰脂质体在mRNA疫苗领域的应用
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【公司研究】键凯科技-深度报告:PEG领域模式创新领先者-210615(27页).pdf
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国防军工PE/PEG估值点阵
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行业数据
2026-07-08
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表9.15 “个体化mRNA肿瘤疫苗”工程开发前沿中核心专利的主要产出国家
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行业数据
2026-03-31
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图37mRNA-LNP疫苗相关良症状分类
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行业数据
2026-03-16
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2025年多个mRNA疫苗产品获得临床批件
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行业数据
2025-12-23
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全球主要PEG
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行业数据
2025-11-19
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美股7巨头与中国科技龙头PEG对比
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行业数据
2025-11-07
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亮丙瑞林微球、布比卡因脂质体、紫杉醇(白蛋白)管线市场情况
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行业数据
2025-11-07
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PCSK9siRNA通过与RISC复合物结合破坏PCSK9mRNA
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行业数据
2025-09-23
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可比公司PEG估值
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2025-09-08
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图表15国证2000、创业板指、北证50近一年PEG变化
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行业数据
2025-08-27
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2022年起,中美科技股的PEG估值开始出现分化
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行业数据
2025-08-27
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三大固态电解质体系及材料特性
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2025-06-27
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完全整合且经过临床验证的AI+mRNA平台
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2025-05-26
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2025年mRNA平台催化剂
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行业数据
2025-05-26
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mRNA与siRNA疗法对比
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2025-05-15
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创新疫苗领域的新应用:PEG 修饰脂质体以强化递送效率,但潜在负面影响值得关注。PEG 修饰被应用于此次新冠疫情中广泛接种的 mRNA 疫苗中,如辉瑞-BioNTech 的BNT162b2,和 Moderna 的 mRNA-1273,前者辅料中采用 ALC-0159(2-[(polyethylene glycol)-2000]-N,N-ditetradecylacetamide),后者辅料中同样包含 PEG 衍生物。此次两款mRNA 疫苗通过 PEG 修饰脂质体强化递送效率,但 PEG 修饰应用的难点在于较广泛出现的 PEG 抗体可能导致不可控的免疫反应和加速血清清除(accelerated blood clearance,ABC)。我们认为,近年来研究较多的核壳型纳米载体中常采用含有 PEG 结构的阴离子聚合物作为外层覆盖物,通过静电相互作用方式包裹在基因复合物颗粒的表面,形成亲水外壳层起到保护核酸的作用,PEG 修饰在核酸药物递送、创新疫苗设计、脂质体强化等领域的应用有望逐步增加。针对可能出现的 PEG 抗原反应、妨碍内吞体妨碍反应等问题,可以通过刺激响应性脱除 PEG(即可断裂 PEG 载体)、氧化还原刺激响应等方式规避,疫苗中的过敏反应机制仍需要进一步研究,PEG 抗原影响可能只是潜在原因之一,我们仍看好 PEG 修饰在新给药平台、给药方式中的应用领域拓展。
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