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图6、BTKPROTAC(P13I)对BTK的降解具有选择性
图6、BTKPROTAC(P13I)对BTK的降解具有选择性
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所属报告:
医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
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METHANOL 在阳光下选择性转化为氢气的国际合作
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2026-03-13
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图10 1985–2015年间,选择的区域走廊内,目的地在发明后五年内重用的来源突破性发明的份额
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竞争格局
2026-03-03
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选择性儿童中枢神经系统肿瘤的发病率和5年总生存率 神经系统肿瘤:2000–2022
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2026-02-13
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“预计2026年的B2B环境将为私募股权提供一个更健康、更可预测的环境,尽管仍会保持选择性。”
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2026-02-13
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图 35 来自欧洲国防、安全和韧性初创公司的选择性收入
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2026-02-12
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奶茶品牌推新中可见中国风味选择的多样性
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行业数据
2026-02-03
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韩国STDP选择性歧化利润
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行业数据
2026-01-20
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韩国STDP选择性歧化利润
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行业数据
2026-01-14
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韩国STDP选择性歧化利润
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行业数据
2026-01-12
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韩国STDP选择性歧化利润
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行业数据
2026-01-07
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BTK抑制剂国内获批情况
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2025-12-31
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韩国STDP选择性歧化利润
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行业数据
2025-12-26
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韩国STDP选择性歧化利润
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行业数据
2025-12-23
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图表17BTKPROTAC全球临床阶段竞争格局
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竞争格局
2025-12-22
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韩国STDP选择性歧化利润
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行业数据
2025-12-19
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行业数据
2026-07-30
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另一方面,由于 PROTAC相关的三元复合物形成需要一定的结构空间,因此原本小分子抑制剂会脱靶(off-target)结合的非靶蛋白,则难以被相应的 PROTAC降解。例如,EGFR小分子抑制剂奥希替尼,则具有约 31个脱靶结合位点;而相应的一种 EGFR PROTAC 分子如 CFT8919特异性降解 EGFR L858R。相似的靶点选择性差异情况也在 BTK小分子抑制剂和 BTK PROTAC之间得到体现,伊布替尼脱靶结合 ITK、EGFR等非靶蛋白,而基于伊布替尼开发的 BTK PROTAC如PI13I,对 BTK具有高度靶点选择性降解能力,而对 EGFR、ITK等非靶靶点不具有降解活性。
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医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
2026年 PROTAC行业报告:BTK PROTAC启动3期,ER降解剂ESR1突变疗效分析|兴业
表9、EGFRPROTAC全球临床阶段竞争格局
表8、ARPROTAC在去势抵抗前列腺癌(CRPC)的临床数据对比
表7、ARPROTAC全球临床阶段竞争格局
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