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全球主要已经上市获批的FGFR抑制剂销售及未来销售预测
全球主要已经上市获批的FGFR抑制剂销售及未来销售预测
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所属报告:
和誉(2256.HK)-港股公司首次覆盖:中国小分子新药研发标兵迎接商业化转型元年-251002(44页).pdf
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图27:iPhone17Pro(256GB)和iPhone7的价格(来自2017年《世界价格地图》版本,完整可用列表,美元)
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行业数据
2026-07-21
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地图来源:自然资源部标准地图服务系统-世界地图,审图号:GS(2016)2945号
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行业数据
2026-07-13
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图8-8:国际武术联合会 《第五届世界太极拳锦标赛竞赛规程》,2026年4月23一30日
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行业数据
2026-07-01
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2000~2025年世界一次能源费结构
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行业数据
2026-07-01
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中国化工产品销售规模占比世界46%(2024年)
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市场规模
2026-07-01
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世界主要运载火箭发射报价(万美元)和运载能力(kg)对比
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行业数据
2026-06-26
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JAK抑制剂在骨髓纤维化治疗中的竞争格局
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竞争格局
2026-06-26
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2026年中国球迷观看往届世界杯时长
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行业数据
2026-06-15
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截至2026年5月4日,美国海军在世界各地部署的航母打击群和两栖戒备群的大致位置
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行业数据
2026-06-12
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中国港口吞吐量世界排名领先,全球TOP10
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行业数据
2026-06-12
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中国港口吞吐量世界排名领先,全球TOP10货
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行业数据
2026-06-12
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图3-1丨世界能源可持续性总分(2022)
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行业数据
2026-06-09
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世界各国家(140个)
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行业数据
2026-06-09
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2025世界能源可持续性评价报告|聚焦全球性冲击影响
fCDpobnnm64gICAgICAgICB8IOWGheWuuSAgICAgICAgICAgICAgICAgICAgIHwKfC0tLS0tLS0tLS0tLS0tfC0tLS0tLS0tLS0tLS0tLS0tLS0tLS0tLS0tfAp8IOaKpeWRiuWQjeensCAgICAgfCAyMDI15LiW55WM6IO95rqQ5Y+v5oyB57ut5oCn6K+E5Lu35oql5ZGKIHwKfCDogZrnhKbkuLvpopggICAgIHwg5YWo55CD5oCn5Yay5Ye75b2x5ZONICAgICAgICAgICB8CgrotYTmlpnmnaXmupDvvJrlm77niYfkuK3mmL7npLrnmoTmlofmnKzkv6Hmga8=
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行业数据
2026-06-09
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世界半导体贸易规模及半导体行业指数均明显上行
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结论:我们认为泛FGFR抑制剂的开发热情将逐渐下降,之前不同公司的pan-FGFR抑制剂的临床开发过程,进一步提升了制药行业对该靶点复杂性及肿瘤特异性的理解。未来更多具备高度选择性的特异性FGFR抑制剂将成为是主流。为了克服由于非选择性抑制剂的脱靶效应引起的并发症,已经开发了第二代FG选 F择R性 TKI,由于该受体家族不同成员的结构同源性,大多数TKI能够靶向一种以上的FGFR。但目前只有少数进入临床试验。与非选择性TKIs相比,这些选择性治疗剂的副作用减少了,最显著的副作用表现为FGF23途径的调节,随之发生钙和磷代谢的改变,如高磷血症和组织钙化。
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和誉(2256.HK)-港股公司首次覆盖:中国小分子新药研发标兵迎接商业化转型元年-251002(44页).pdf
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和誉截至2025年9月的临床管线示意
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