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图17、MAT2A抑制剂与PRMT5抑制剂具有协同效应
图17、MAT2A抑制剂与PRMT5抑制剂具有协同效应
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所属报告:
百济神州-公司研究报告-临床早期差异化管线布局丰富助推长期快速发展-250723(50页).pdf
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JAK抑制剂在骨髓纤维化治疗中的竞争格局
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竞争格局
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《KAT6抑制剂化合物、药物组合物及其制备方法和N-(6-((1H-pyrazol-1-yl)methyl)-4-metho
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行业数据
2026-05-11
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图10、全球PD-(L)1抑制剂市场规模(十亿美元)
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市场规模
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①内部四大业务板块协同的规模效应
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市场规模
2026-04-27
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图10.VMAT2抑制剂全球销售情况(亿美元)
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行业数据
2026-04-20
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全球PCSK9抑制剂市场规模(亿美元)
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市场规模
2026-04-13
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中国PCSK9抑制剂市场规模(亿人民币)
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市场规模
2026-04-13
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相较于PD-(L)1抑制剂,PD-(L)1/VEGF双抗有极大替代和拓展空间
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行业数据
2026-03-31
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全球在研FXI/FXIa抑制剂的临床进展
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行业数据
2026-02-26
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FXI/FXIa抑制剂全球可触及患者数
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行业数据
2026-02-26
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图表11FDA获批KRASG12C抑制剂的全球销售额(百万美元)
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行业数据
2026-02-25
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图表19KRASG12D抑制剂竞争格局
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竞争格局
2026-02-25
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图3 mCRC中EGFR抑制剂的美国收入(2004-2017)
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行业数据
2026-02-13
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主要JAK抑制剂全球销售额
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行业数据
2026-01-30
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国内主要JAK抑制剂在研格局
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2026-01-30
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MAT2A 抑制剂与 PRMT5 抑制剂具有协同效应,可以通过联用方案,提高对于MTAP 缺失肿瘤的治疗效果。在 PRMT5/MTAP“( 合成致死”组合中,MAT2A 蛋白也是重要的参与成员:由于 MTAP 缺失突变后,大量积累的 MTA 与 PRMT5 正常的底物 SAM 具有竞争性,从而抑制 PRMT5 正常的甲基化功能;而 MAT2A 酶主要用于产生 SAM,因此通过进一步抑制 MAT2A 可以从源头阻断 SAM 合成,提高 PRMT5/MTAP“合成致死”的效果。
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百济神州-公司研究报告-临床早期差异化管线布局丰富助推长期快速发展-250723(50页).pdf
表9、CDK2选择性抑制剂的全球竞争格局(临床阶段)
表8、CDK4选择性抑制剂的全球竞争格局(临床阶段)
表7、BGB-43395与CDK4、CDK4/6抑制剂在治疗2L+ER+乳腺癌的临床数据对比(非头对头对比)
表6、海外MNC药企在HR阳性乳腺癌的产品管线布局
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