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公司JJH201501及JJH201601新药项目实施阶段
公司JJH201501及JJH201601新药项目实施阶段
行业数据
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图片大小:288KB
图片尺寸:2303*706
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所属报告:
吉贝尔-核心产品赋能成长业绩有望加速释放-221216(18页).pdf
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JJH201501和对照药物的临床药代动力学参数对比
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多西他赛衍生物药效显著提高且毒副作用明显降低。多西他赛衍生物(JJH201601)是公司依托脂质体药物研发技术平台开发的一类在研抗肿瘤新药。公司和上海交通大学颜德岳院士团队对多西他赛进行结构改造,通过分子设计和药效试验筛选得到全新化合物JJH201601,利用脂质体技术将其开发为脂质体制剂。目前已完成临床前试验研究,结果显示与多西他赛相比疗效显著,裸鼠模型药效显著提高且毒副作用明显降低,抑瘤率超 99%,且停药后观察期内未发现肿瘤复发,该结果在肺癌 A549、肝癌 HepG2 和胰腺癌 Panc-1模型均得以验证。目前 JJH201601准备提交临床试验申请,据公司综合测算上市后 3-5年内年收入规模有望突破 5亿元。
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吉贝尔-核心产品赋能成长业绩有望加速释放-221216(18页).pdf
JJH201501和对照药物的临床药代动力学参数对比
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