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图13、Vepdegestrant+哌柏西利临床1b期试验中期结果及与同类方案数据对比(非头对头数据)
图13、Vepdegestrant+哌柏西利临床1b期试验中期结果及与同类方案数据对比(非头对头数据)
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图片大小:479KB
图片尺寸:2221*1149
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所属报告:
医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
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图表48哌柏西利、瑞波西利、阿贝西利结构及主要副
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行业数据
2025-02-24
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图表51哌柏西利、瑞波西利、阿贝西利全球销售额/亿
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行业数据
2025-02-24
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哌柏西利、阿贝西利、利柏西利和达尔西利治疗晚期乳腺癌疗效对比分析
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行业数据
2023-03-15
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表6、CDK4/6抑制剂国内样本医院销售额(百万元)202020212022哌柏西利13.1824.469.65
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行业数据
2023-03-15
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阿贝西利与派柏西利用于晚期乳腺癌治疗对比
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联用方面,Vepdegestrant探索与 CDK4哌柏西利联合用药。Arvinas于 ESMO BC 2024公开 ARV-471联用哌柏西利(CDK4)的临床 1b期更新结果,对于既往接受过中位 4 线治疗的 ER+/HER2-乳腺癌患者,ARV-471 联合哌柏西利在mPFS实现 11.2个月( 其中 ESR1突变患者中为 13.7个月);安全性方面,3级或 4级治疗相关的中性粒细胞减少为 91%、白细胞降低为 15%,预计可以通过哌柏西利减量实现改善。
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医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
2026年 PROTAC行业报告:BTK PROTAC启动3期,ER降解剂ESR1突变疗效分析|兴业
表9、EGFRPROTAC全球临床阶段竞争格局
表8、ARPROTAC在去势抵抗前列腺癌(CRPC)的临床数据对比
表7、ARPROTAC全球临床阶段竞争格局
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