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图19.多奈哌齐和氟诺哌齐(DC20)分子结构
图19.多奈哌齐和氟诺哌齐(DC20)分子结构
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康缘药业(600557)-A股公司研究报告:“一体两翼”战略价值凸显创新布局未来可期-250804(24页).pdf
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图17、SAR444200分子结构
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行业数据
2026-02-04
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中国分子诊断市场应用结构
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行业数据
2026-01-26
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图68WO2021092266A1利文披露的GNC台多抗分子结构
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行业数据
2025-12-23
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图67WO2023246885A1利DLL3xCD3特性结合蛋白分子结构
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行业数据
2025-12-23
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Lp(a)的分子结构示意图以及不同脂蛋白(VLDL/IDL/LDL)之间的相互转化
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行业数据
2025-11-20
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自然堂集团细分子渠道收入结构(单位:亿元)
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行业数据
2025-11-07
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Lp(a)小分子抑制剂结构示意图
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行业数据
2025-11-05
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ZL-1310(DLL3ADC)分子结构
fCDnu4Tku7YgfCDmj4/ov7AgfAp8IC0tLS0gfCAtLS0tIHwKfCBBIHwg5Lq65rqQ5YyW5oqXIERMTDMgSWdHMSDljZXlhYvpmobmipfkvZMgfAp8IEIgfCDlj6/oo4Lop6PkuInogr3ov57mjqXlrZAgfAp8IEMgfCDllpzmoJHnorHooY3nlJ/nianmnInmlYjovb3ojbfvvIhDMjQg5Z6L77yJ77yM6I2v54mp5oqX5L2T5q+U77yIREFS77yJPTggfAoK6LWE5paZ5p2l5rqQ77ya5YaN6byO5Yy76I2vIDJRMjUgUFBU77yM55Sz5LiH5a6P5rqQ56CU56m2
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行业数据
2025-09-24
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7MW4911的分子结构
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行业数据
2025-09-08
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多奈哌齐片剂2018-2022国内医院终端
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行业数据
2025-08-08
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CS2009分子结构设计
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行业数据
2025-08-06
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图21.DC20在老年受试者单次给药后的主要药代动力学参数
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行业数据
2025-08-05
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图20.氟诺哌齐一期临床设计
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2025-08-05
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2025-07-28
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公司联合中科院上海药物所开发的氟诺哌齐(DC20)是一种新型乙酰胆碱酯酶抑制剂,开发思路主要是基于多奈哌齐的结构,在其哌啶环和苄基苯环部分引入氟原子进行改造而获得。相比多奈哌齐,氟诺哌齐的临床前药效研究显示,其基于与乙酰胆碱酯酶的高亲和力和慢解离的特点,对乙酰胆碱酯酶的抑制效果更强,约为多奈哌齐的 6倍,且选择性(抑制乙酰胆碱酯酶的 IC50值与抑制丁酰胆碱酯酶的 IC50值的比值)更高,为多奈哌齐的 6.8 倍,此外,DC20 在小鼠大脑以及大鼠大脑皮层和海马体中的效力分别比多奈哌齐体外抗 AChE活性强 3倍、16倍和 8倍,表明氟诺哌齐的靶点选择性和抗 AChE活性更好。
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