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口服SERD针对CDK4/6i经治及ESR1突变人群疗效优异,有望成为新一代内分泌疗法
口服SERD针对CDK4/6i经治及ESR1突变人群疗效优异,有望成为新一代内分泌疗法
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所属报告:
肿瘤创新药行业首次覆盖:抗肿瘤疗法持续迭代国产新药迎来突破-250313(66页).pdf
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行业数据
2026-01-28
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2025Q4新一代信息技术领域招聘TOP5城市
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行业数据
2026-01-19
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2025Q4新一代信息技术领域增长亮眼的职业
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行业数据
2026-01-19
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自动驾驶出行市场生态构成图(主要基于Robotaxi方案提供商的最新一代车型)
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行业数据
2026-01-12
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第一代EGFR-TKI不同企业竞争格局
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竞争格局
2026-01-08
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AIEV(人工智能电动汽车)是指以电动化为基础、网联化为支撑、AI为核心的新一代智能汽车,通过智能驾驶、智能座舱、智能底盘等技术的深度融合及软硬协同,
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行业数据
2025-12-24
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行业数据
2025-12-15
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口服 SERD 等新兴疗法有望提供更优的内分泌治疗方案。现行内分泌药物包括他莫昔芬、雌激素受体调节剂、芳香化酶抑制剂(AI)、氟维司群等。目前芳香化酶抑制剂为最主流的基石疗法。选择性雌激素受体降解剂(SERD)可通过诱导 ER 降解,切断乳腺癌细胞生长信号,氟维司群为全球首款 SERD 药物,但分子量较大、口服生物利用度低,使其仅能通过肌肉注射给药,患者依从性差。近年来,口服 SERD 药物成为新一代内分泌疗法的研发重点之一,具体的开发路径包括:(1)联合 CDK4/6 抑制剂,用于 HR+HER2-乳腺癌的一线治疗,目前阿斯利康、罗氏在全球进展领先;(2)单药用于 HR+HER2-乳腺癌的二线治疗,Radius 的 Elacestrant 已在海外获批,国内益方生物的 Taragarestrant 处于 III 期临床、进展领先。在疗效方面,口服 SERD 针对 CDK4/6i 经治及 ESR1 突变人群疗效尤其优异。
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肿瘤创新药行业首次覆盖:抗肿瘤疗法持续迭代国产新药迎来突破-250313(66页).pdf
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