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维迪西妥、T-DM1和DS-8201结构对比
维迪西妥、T-DM1和DS-8201结构对比
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所属报告:
荣昌生物-公司深度报告:ADC+自免双驱期待国际化突破-240326(30页).pdf
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维迪西妥单抗联合免疫奠定在HER2表达mUC患者晚期一线治疗的标准治疗地位(非头对头)
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行业数据
2025-10-23
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主要注射型GLP-1药物减重临床数据对比(非头对头,调整PBO,非T2DM人群)
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行业数据
2025-09-18
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使用维迪西妥单抗(RC48)2.0mg/kg治疗的患者周围
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行业数据
2025-06-27
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T-DXd快速抢占T-DM1美国市场份额,同时全球市场份额保持高位
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竞争格局
2025-06-03
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2021-2024Q1年维迪西妥单抗收入(百万元)
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其它
2024-07-11
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维迪西妥临床管线丰富
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2024-03-29
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维迪西妥国内销售额测算
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2024-03-29
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表7、DS8201与T-DM1设计对比
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2024-02-28
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2022年1月-2023年6月唐DM月度销量
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2023-08-21
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DS-8201拥有比T-DM1更高的稳定性和均一性
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2023-07-21
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在小鼠肿瘤模型中,ZW49表现出比T-DM1和DS-8201更强的抗肿瘤活性
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2023-05-23
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2026-07-30
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1)旁杀效应较为突出。采用优化后可酶切的连接子,基于“旁杀效应”提高对肿瘤组织的整体杀灭效果,同时提高 ADC 药物的血液稳定性和安全性。维迪西妥单抗的可酶切连接子在被肿瘤细胞内吞且经酶切消化后,释放的连接子-细胞毒素复合物分子量较小、具备较高的膜通透性,从而可以逸散至附近的其他肿瘤细胞(包括 HER2 不表达的细胞),带来较好的“旁杀效应”。T-DM1 连接子降解后释放的连接子-细胞毒素复合物分子量较大、具备较低的膜通透性和“旁杀效应”。
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