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国内全身麻醉镇静药在研情况
国内全身麻醉镇静药在研情况
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所属报告:
海思科(002653)-A股公司研究报告:创新转型成效显著多款新药上市放量-250929(48页).pdf
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环泊酚的比较优势突出,市场竞争格局较好。与丙泊酚相比,在手术室外麻醉领域:环泊酚具有起效迅速、苏醒快速、镇静成功率 100%、更少呼吸抑制、更少注射痛,发生率仅为丙泊酚 1/10,效价为丙泊酚 4-5 倍、更少用量,安全窗更宽、更少操作,使用更便捷、总体不良事件发生率更低等优点;在手术室内麻醉领域:环泊酚具有起效迅速、苏醒快速、镇静成功率 100%、维持期间 BIS 曲线更平稳、更少心血管不良事件、循环平稳、更少注射痛,提高患者舒适度、效价为丙泊酚 4-5 倍,更少用量,安全窗更宽、总体不良事件发生率更低等优点。目前,国内已获批上市的镇静新药主要有 4 款,分别为海思科的环泊酚、恒瑞医药的甲苯磺酸瑞马唑仑、宜昌人福的苯磺酸瑞马唑仑及磷丙泊酚二钠。相比于其他镇静新药,环泊酚具有获批适应症广、剂型(乳剂)便利性高等优势。国内在研的全身麻醉镇静药较少,其中恩华药业的 NH600001 乳状注射液已完成 III 期临床阶段,预计 2025 年申报 NDA。
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海思科(002653)-A股公司研究报告:创新转型成效显著多款新药上市放量-250929(48页).pdf
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国内全身麻醉镇静药在研情况
国内近年获批上市的镇静新药
海思科主要的仿制药品种
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