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主要癌症PIK3突变几率
主要癌症PIK3突变几率
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所属报告:
翰森制药-港股公司研究报告-深入布局优质赛道创新升级赋能新里程-230316(35页).pdf
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相关数据
图表28PIK3CA靶点产品的竞争格局
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2024-04-23
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1)乳腺癌药物需求广阔:根据国家癌症中心发布的 2022 年癌症报告,2016 年乳腺癌新发病例总数在主要癌症中排名第四,因此乳腺癌药物需求广阔。2)PIK3 抑制剂适用患者较多:公司 HS-10352 针对的靶点 PIK3 在乳腺癌患者中突变率高达 26.0%,适用患者较多。3)临床数据表明公司产品的疗效与安全性良好:根据公司在美国癌症研究协会(AACR)会议发布的 1 期临床数据,6 例 PIK3CA 突变患者中,ORR 为50.0%,9 个月无进展生存率(PFS 率)为 66.7%,有效性良好。安全性层面,18 例患者中仅两例发生较为严重的副作用(3 级高血糖),发生皮疹的患者为两例。相对比,全球首个获批的 PIK3 抑制剂诺华(NVS US)的 Alpelisib+氟维司群组在临床试验中表现出的客观缓解率(ORR)为 35.7%,PFS 为 9.1 个月,3-4 级皮疹与高血糖发生率分别为 20%与 33%。虽然 1 期临床病例数量较少并不能反映最终结果,但是从以上数据看 HS-10352 没有表现出劣势。4)目前国内还没有其他针对 PIK3 靶点药物获批,因此 HS-10352 如能成功上市,先发优势很强。目前全球获批用于乳腺癌治疗的同靶点产品仅诺华(NVS US)的Alpelisib,并且没有进入中国,因此如公司产品能顺利上市,先发优势明显。
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当前图表所属:
翰森制药-港股公司研究报告-深入布局优质赛道创新升级赋能新里程-230316(35页).pdf
三代EGFR-TKI制剂对比
2016年国内主要癌症新发病例数量(单位:万人)
公司肿瘤领域主要仿制药市场份额
:财务摘要(年结:12月31日;人民币百万元)
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