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图19、IRAK-4参与TLRs/IL-1R信号通路
图19、IRAK-4参与TLRs/IL-1R信号通路
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图片大小:991KB
图片尺寸:1749*1190
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所属报告:
医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
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(五)IRAK4:自免领域潜力巨大,有望打破该靶点上市药物空白局面 IRAK4 在炎症性疾病的发病和进展发挥重要作用。IRAK(白细胞介素 1 受体相关激酶 4)作为在 Toll 样受体(TLR)及白介素-1 受体(IL-1R)介导的信号通路的重要连接体,在炎症相关信号通路中发挥重要作用。研究表明 IRAKs参与了炎症性肠病、酒精性肝病、炎症相关性结直肠肿瘤等消化系统疾病的发生发展。在激活TLR/IL1R后,TLR胞内募集适配蛋白 IRAK4/2,IRAK4通过激活 IRAK1,进而在下游激活一系列转录因子(NF-κB等),促进促炎症细胞因子分泌,免疫细胞增殖分化等。目前,尚无靶向 IRAK4 的药物上市,但研究表明靶向 IRAK4 在炎症及 B细胞淋巴瘤中发挥着关键作用。
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医药生物行业PROTAC深度报告:探索“不可成药难题”的解决方案拓展肿瘤、自身免疫等领域市场潜力-250522(37页).pdf
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